Cell Line | Cell Type | HER2/neua | PI-9b | IC50 (nM) | ||
---|---|---|---|---|---|---|
GrB | GrB-Fc-4D5 | Kadcyla | ||||
Calu-3 | Lung | 109 | 0.5 | > 1000 | 82 | 0.02 |
SKBR3 | Breast | 100 | 48 | > 1000 | 56 | 0.02 |
NCI-N87 | Gastric | 85 | 8 | > 1000 | 105 | 139 |
MDA-MB-453 | Breast | 13 | 0.4 | 532 | 32 | 0.55 |
SKOV3 | Ovarian | 11 | 100 | > 1000 | 211 | 38 |
DU-145 | Prostate | 3.6 | 3 | > 1000 | 45 | 152 |
MCF-7 | Breast | 3.4 | 38 | > 1000 | 99 | 24 |
SKMEL28 | Melanoma | 3.4 | 73 | > 1000 | 67 | 63 |
HT-29 | Colon | 3.0 | 0.6 | > 1000 | 36 | 39 |
A-549 | Lung | 2.4 | 31 | > 1000 | 55 | 78 |
MDA-MB-231 | Breast | 1.5 | 79 | 793 | 27 | 44 |
A375-M | Melanoma | 1.5 | 27 | > 1000 | 28 | 28 |
AAB-527 | Melanoma | 1.3 | 39 | > 1000 | 57 | 25 |
MDA-MB-468 | Breast | 1.1 | ND | > 1000 | 64 | 31 |