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Table 4 Druggable sites identified by SiteMap

From: KLF7: a new candidate biomarker and therapeutic target for high-grade serous ovarian cancer

 

SiteScore

Residues

Site1

0.866

Gly225, Cys226, Arg227, Lys228, Val229, Tyr230, Hys235, Ala238, Hys239, Thr242, Hys243, Pro248, Tyr249, Lys250, Cys251, Ser252, Trp253, Glu254, Gly255, Cys256, Glu257, Trp258, Arg259, Ser263, Asp264, Leu266, Thr267, Tyr270, Arg271, Thr274, Ala276.

Site2

0.838

Trp258, Phe260, Ala261, Glu265, Arg268, Hys269, Arg271, Lys272, Gly275, Ala276, Lys277, Phe288, Ser289, Arg290, Hys293.

Site3

0.812

His219, Arg220, Cys221, Gln222, Phe223, Ser233, Leu236, Lys237, Gln240, Arg241, His243, Thr244