Tumor model | TGI (%) | RESPONSE at 1.9 mg/Kg | ||
---|---|---|---|---|
ORR (%) | ||||
Genz-644282 | The-0504 | Genz-644282a | The-0504 | |
Pancreatic (PaCa44) | 64.2 | 100 | 33.3% SD | 100% MCR |
16.7 | 100 | 66.7% PD | ||
Colorectal (HT29) | Not available | Not available | 33.3% SD | 66.7% CR |
16.6 | 100 | 66.7% PD | 33.3% PR | |
Breast (MDA-MB 231) | 70.1 | 100 | 16.7% SD | 83.3% MCR |
0 | 100 | 83.3% PD | 16.7% CR | |
Liver (HepG2) | 55.5 | 100 | 25.0% PR | 100% MCR |
25.0 | 100 | 75.0% PD | ||
Pancreatic (PDX)a | 0 | 93.6 | 100% PD | 33.3% MCR |
0 | 83.3 | 16.7% CR, | ||
33.3% PR, | ||||
16.7% SD |