Agents | Cancer | Cell Type | Combined | Ref |
---|---|---|---|---|
A1210477 | AML | THP-1 U937 | venetoclax | [337] |
A1210477 | Breast | MDA-MB-231 cells | TRAIL | [338] |
A1210477 | Cervical | SiHa and CaSki | navitoclax | [139] |
A1210477 | CML | K562, K562/R | EE-84 | [339] |
A1210477 | CRC | RKO, HT29, A375 | cobimetinib | [340] |
A1210477 | DLBCL | U-2946 | navitoclax | [341] |
A1210477 | PC, GC, NSCLC, MM | BxPC-3, EJ-1, H23, and OPM-2 | navitoclax | [70] |
A1210477 | HNSCC | PCI15B, Detroit 562, MDA686LN, and HN30 | navitoclax | [342] |
A1210477 | nHL | SU-DHL-4, WSU-NHL, WSU-DLCL2, KARPAS-422 | venetoclax | [343] |
AMG-176 | CLL | Patient samples (5) | venetoclax | [344] |
AZD-5991 | AML | OCI-AML3 and MCL-1-OE Molm13 and MV4–11 | venetoclax | [345] |
AZD5991 | MM | NCI-H929 | bortezomib, venetoclax | [73] |
GDC-0941 | Breast | MDA-MB-231, SKBR3 | ABT-737 | [346] |
Mim1 | Glioblastoma | U87mg | temozolomide | [347] |
Mim1 | Melanoma | C32 melanoma cells | dacarbazine | [348] |
Mim1 | MM | Colo829 | dacarbazine | [349] |
S63845 | AML | OCI-AML3, MOLM-13, OCI-AML2 | trametinib/HDM201 | [350] |
S63845 | AML | Primary samples | venetoclax | [351] |
S63845 | AML | MOML-13, SKM-1, | trametinib | [352] |
S63845 | AML | Cell lines and primary cells | venetoclax | [353] |
S63845 | Breast | SK-BR-3 | docetaxel, trastuzumab, lapatinib | [354] |
S63845 | CRC | HCT116 | regorafenib | [355] |
S63845 | Mantle cell lymphoma | Patient-derived xenografts | venetoclax | [356] |
S63845 | Melanoma | Patient samples | navitoclax | [357] |
S63845 | Melanoma | MeWo | TRAIL resistance | [358] |
S63845 | Myeloma | U266 xenograft | venetoclax | [359] |
S63845 | MM | MOL-P8, OPM-2, NCI-H929 | venetoclax, bortezomib | [360] |
S63845 | MM | RPMI-8226 xenograft | venetoclax | [361] |
S63845 | Nasopharyngeal carcinoma | CNE-2, 5-8F | venetoclax | [293] |
S63845 | T-ALL | Zebrafish T-ALL cells | venetoclax | [304] |
VU661013 | AML | MV-4-11, AML-001/2, patient xenografts | venetoclax | [76] |
VU661013 | Breast | HCC1428, MCF7, T47D | navitoclax | [362] |